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Bio
许叶春研究员及其课题组主要开展基于靶标结构的药物设计研究,建立了以精准表征化合物与靶标结合为特色的多学科交叉、多技术整合的先导化合物从头设计与高效优化研究策略与技术体系,针对感染与炎症密切相关的重要蛋白质,快速发现活性化合物,解析多个关键化合物与靶标结合的高分辨率复合物结构,并精确测定化合物与靶标的亲和力,从而精准表征化合物与靶标结合的位点、相互作用模式、构象变化、水分子的作用及热力学特征等,同时应用计算机辅助药物设计方法,高效获得了多个全新先导化合物及临床前、临床候选新药。
Research Interests
Papers共 192 篇Author StatisticsCo-AuthorSimilar Experts
By YearBy Citation主题筛选期刊级别筛选合作者筛选合作机构筛选
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Yan Zhong, Li Shi, Zhuo Xu,Jing Gao, Qingyu Ma, Tianqi Gao, Junying Tang, Muya Xiong,Yechun Xu, Huixiong Dai,Hu Zhou,Naixia Zhang, Chen Zhou
Communications biologyno. 1 (2025): 761-761
Wenfeng Zhao,Guofeng Chen, Jian He, Xiaofang Shen, Muya Xiong, Liwei Xiong, Zhihao Qi,Hang Xie, Wanchen Li, Jiameng Li, Huixia Dou, Hangchen Hu, Haixia Su,Qiang Shao,Minjun Li,Hongbin Sun,Yechun Xu
Nature communicationsno. 1 (2025): 5140-5140
Haixia Su,Guofeng Chen,Hang Xie, Wanchen Li, Muya Xiong, Jian He, Hangchen Hu, Wenfeng Zhao,Qiang Shao,Minjun Li,Qiang Zhao,Yechun Xu
Nature communicationsno. 1 (2025): 4288-4288
Bioorganic chemistry (2025): 108503-108503
Haixia Su, Guoqing Wu, Muya Xiong, Yuhang Wang, Junyuan Cao, Mengyuan You, Yingchun Xiang, Tianqing Nie,Minjun Li,Gengfu Xiao,Leike Zhang,Qiang Shao,Yechun Xu
Advanced science (Weinheim, Baden-Wurttemberg, Germany)pp.e2501625-e2501625, (2025)
Shulei Hu,Yumin Zhang, Chenchen Wang,Jian Li, Haixia Su, Xiong Xie,Jiang Wang, Jinlin Wang, Junyuan Cao, Xiaofei He,Yechun Xu,Leike Zhang, Wenhao Dai,Hong Liu
Journal of medicinal chemistryno. 11 (2025): 10823-10844
STEROIDS (2024)
J Chem Inf Modelno. 24 (2024): 9501-9516
Wang Xudong, Xiong Liwei, Zhu Ying,Liu Sixiu,Zhao Wenfeng,Wu Xinyuan, Seydimemet Mengnisa,Li Linjie, Ding Peiqi, Lin Xian,Liu Jiaxiang, Wang Xuan,Duan Zhiqiang,Lu Weiwei,Suo Yanrui, Cui Mengqing,Yue Jinfeng,Jin Rui,Zheng Mingyue,Xu Yechun, Mei Lianghe,Hu Hangchen,Lu Xiaojie
chinaxiv(2024)
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Ying Qin,Dekang Li,Chunting Qi,Huaijiang Xiang,Huyan Meng,Jingli Liu,Shaoqing Zhou,Xinyu Gong,Ying Li, Guifang Xu,Rui Zu,Hang Xie,Yechun Xu, Gang Xu,Zheng Zhang, Shi Chen,Lifeng Pan,Li Tan
ACTA PHARMACEUTICA SINICA Bno. 1 (2024): 319-334
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Author Statistics
#Papers: 192
#Citation: 13370
H-Index: 46
G-Index: 114
Sociability: 7
Diversity: 3
Activity: 80
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