Discovery of a Potent and Highly Selective PDK1 Inhibitor Via Fragment-Based Drug Discovery.
Bioorganic & Medicinal Chemistry Letters(2011)
关键词
PDK1,Selective,Tethering,Pyridinone,DFG-out,Fragment-based drug discovery
AI 理解论文
溯源树
样例

生成溯源树,研究论文发展脉络
Chat Paper
正在生成论文摘要