A Three-Step Protocol for Lead Optimization: Quick Identification of Key Conformational Features and Functional Groups in the SAR Studies of Non-Atp Competitive MK2 (MAPKAPK2) Inhibitors
Bioorganic & Medicinal Chemistry Letters(2012)
关键词
Three-step protocol,SAR,Conformation,MK2,TNF alpha,Non-ATP competitive,Inhibitor
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