Development of the Large-Scale Synthesis of Tetrahydropyran Glycine, a Precursor to the HCV NS5A Inhibitor BMS-986097
Arvind Mathur,Bei Wang,Daniel Smith,Jianqing Li,Joseph Pawluczyk,Jung-Hui Sun,Michael Kwok Wong,Subramaniam Krishnananthan,Dauh-Rurng Wu,Dawn Sun,Peng Li,Shiuhang Yip,Bang-Chi Chen,Phil S. Baran,Qi Chen,Omar D. Lopez, Zhong Yong,John A. Bender,Van N. Nguyen,Jeffrey L. Romine,Denis R. St Lauren,Gan Wang,John F. Kadow,Nicholas A. Meanwell,Makonen Belema,Rulin Zhao JOURNAL OF ORGANIC CHEMISTRY(2017)
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