Aligning Potency and Pharmacokinetic Properties for Pyridine-Based NCINIs.
Lee D. Fader,Murray Bailey,Eric Beaulieu,Francois Bilodeau,Pierre Bonneau,Yves Bousquet,Rebekah J. Carson,Catherine Chabot,Rene Coulombe,Jianmin Duan,Craig Fenwick,Michel Garneau,Ted Halmos,Araz Jakalian,Clint James,Stephen H. Kawai,Serge Landry,Steven R. LaPlante,Stephen W. Mason,Sebastien Morin,Nathalie Rioux,Bruno Simoneau,Simon Surprenant,Bounkham Thavonekham,Carl Thibeault,Thao Trinh,Youla Tsantrizos, Jennifer Tsoung,Christiane Yoakim,Dominik Wernic ACS Medicinal Chemistry Letters(2016)
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HIV integrase,NCINI,enterohepatic recirculation
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