Discovery of E7766: A Representative of a Novel Class of Macrocycle-Bridged STING Agonists (mbsas) with Superior Potency and Pan-Genotypic Activity
Atsushi Endo,Dae-Shik Kim,Kuan-Chun Huang,Ming-Hong Hao,Steven Mathieu,Hyeong-wook Choi,Utpal Majumder,Xiaojie Zhu,Yongchun Shen,Kristen Sanders,Thomas Noland,Dinesh Chandra,Yu Chen,Karen TenDyke,Kara Loiacono,Donna Kolber-Simonds,Rongrong Jiang,Vaishali Dixit,Janna Hutz,John Wang,Xingfeng Bao,Francis Fang,Nadeem Sarwar CANCER RESEARCH(2019)
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transcriptional control,cGAS-STING Pathway
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