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Structure-based Design, Synthesis and Bioactivity Evaluation of Macrocyclic Inhibitors of Mutant Isocitrate Dehydrogenase 2 (IDH2) Displaying Activity in Acute Myeloid Leukemia Cells.

European Journal of Medicinal Chemistry(2020)

引用 5|浏览78
关键词
Metabolic pathways,Isocitrate dehydrogenase 2,Conformational restriction,Macrocyclic derivatives,Inhibitors
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