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P-glycoprotein Substrate Assessment in Drug Discovery: Application of Modeling to Bridge Differential Protein Expression Across in Vitro Tools.

Journal of Pharmaceutical Sciences(2020)

引用 5|浏览20
关键词
Drug transporter,P-glycoprotein,MDR1,P-gp expression,Kinetics,In vitro models,Efflux,Blood brain barrier,MDCK cells
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