Structure-Based Design and Development of Phosphine Oxides As a Novel Chemotype for Antibiotics That Dysregulate Bacterial ClpP Proteases.
Journal of Medicinal Chemistry(2024)
关键词
ClpP,antibiotics,dysregulation,Neisseria meningitidis,Neisseria gonorrhoeae,acyldepsipeptides (ADEPs),activators of self-compartmentalizing proteases (ACPs)
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