Evolution Of Nonbasic Thienopyrimidinone Containing Alcohols As Selective Mchr1 Antagonists Culminating In The Discovery Of The Clinical Candidate Bms-830216 William N. Washburn , Mark Manfredi , Pratik Devasthale , Guohua Zhao , Saleem Ahmad , Andres Hernandez , Jeffrey A. Robl , Wei Wang , James Mignone , Zhenghua Wang , Khehyong Ngu , Mary Ann Pelleymounter , Daniel Longhi , Ning Huang , Neil Flynn , Anthony V. Azzara , Joel C. Barrish , Kenneth Rohrbach , James Devenny , Suzanne Rooney , Michael Thomas , Susan Glick , Helen Godonis , Susan Harvey , Mary Jane Cullen , Simeon Taylor , Hongwei Zhang , Christian Caporuscio , Paul Stetsko , Mary Grubb , Brad D. Maxwell , Hong Yang , Atsu Apedo , Brian Gemzik , Evan Janovitch , Christine Huang , Lisa Zhang , Chris Freeden , Brian J. Murphy ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY(2012)
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