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Asymmetric Synthesis of the Cyclohexyl Fragment in RORγt Inhibitor (BMS-986251) Enabled by a Dynamic Kinetic Resolution of Hageman’s Ester

ORGANIC PROCESS RESEARCH & DEVELOPMENT(2022)

引用 3|浏览15
关键词
DKR,hydrogenation,carbonylation enol nonglatc,directed hydrogenation
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