Fragment-Based Discovery and Structure-Guided Optimization of 2-Benzoyl-7-azabenzimidazoles As Potent, Highly Selective and Orally Active CDK4/6 Inhibitors Young Cho , Christopher Brain , Christine Chen , Hong Cheng , Rajiv Chopra , J. Giraldes , Steven Kovats , Bharat Lagu , Michael J. Luzzio , Junqing Shen , Fan Yang , Wojciech Wrona , Marc O’Reilly , Steven Howard , Alice Loo , Kristy Haas , Sunkyu Kim , Yipin Lu , Wieslawa Maniara , Troy Smith , Mei Ying Xu , Hayley C. Angove , R.K. Cheng , Miles Congreve , Claudio Dagostin , Deborah Davis , Ruth E. Feltell , Steven D. Hiscock , Kim Lewry , Rachel McMenamin , Paul N. Mortenson , Rajdeep K. Benning , David C. Rees , Glyn Williams , Alison J.‐A. Woolford openalex(2012)
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