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Lead Change of a HIF-2α Antagonist Guided by Multiparameter Optimization and Utilization of an O Lp →π* Ar Interaction

MEDICINAL CHEMISTRY RESEARCH(2023)

引用 2|浏览3
关键词
HIF-2α,n→π*,Transcription factor inhibition,Structure based drug design,PT2977,MK-6482
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