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Abstract B137: Selective Inhibition of the Active State of KRASG12V with the Non-Covalent, Tri-Complex Inhibitor RM-048

Bianca J Lee,Jim Cregg, Anne Edwards, Jerry Chen, Andre Eriksson, Emily Tonogai,Aidan Tomlinson,Kyle Seamon, Mariela Moreno Ayala,Nataliya Tovbis Shifrin,Nilufar Montazer, Kate Sanders, Jun Huang,Kang-Jye Chou, Benjamin Madej, Yang Liu,Zhican Wang,Zhengping Wang,John Knox,Elena Koltun,Jingjing Jiang,Adrian Gill,Jacqueline A.M. Smith

Molecular Cancer Therapeutics(2023)

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