Development of Potent Mcl-1 Inhibitors: Structural Investigations on Macrocycles Originating from a DNA-Encoded Chemical Library Screen.
Koen F. W. Hekking,Sergio Maroto, Kees van Kekem, Frank S. Haasjes,Jack C. Slootweg, Patrick G. B. Oude Alink, Ron Dirks,Malvika Sardana, Marjon G. Bolster, Brian Kuijpers, Dennis Smith, Robin Doodeman,Marcel Scheepstra,Birgit Zech,Mark Mulvihill,Louis M. Renzetti,Lee Babiss,Paolo A. Centrella,Matthew A. Clark,John W. Cuozzo,Marie-Aude Guie,Eric Sigel,Sevan Habeshian,Christopher D. Hupp,Julie Liu,Heather A. Thomson,Ying Zhang,Anthony D. Keefe, Gerhard Muller, Stijn Gremmen Journal of Medicinal Chemistry(2024)
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