Iridium-Catalyzed Asymmetric Hydrogenation of Heteroaromatics with Multiple N Atoms Via Substrate Activation: an Entry to 4,5,6,7-Tetrahydropyrazolo[1,5-a]pyrimidine-3-carbonitrile Core of a Potent BTK Inhibitor.
JOURNAL OF ORGANIC CHEMISTRY(2024)
关键词
Asymmetric Catalysis,Selective Hydrogenation,Hydrogenation,Dehydrogenation
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