Abstract GS03-10: Allosteric PI3K-alpha Inhibition Overcomes On-Target Resistance to Orthosteric Inhibitors Mediated by Secondary PIK3CA Mutations
Andreas Varkaris,Ferran Fece de la Cruz,Elizabeth Martin, Bryanna Nordern,Nicholas Chevalier,Ignaty Leshchiner,Anastasia Stavridi,Janice Kim,Alkistis Papatheodoridi,Hakan Gunaydin,Brian Danysh,Laxmi Parida,Ioannis Sanidas,Yongli Ji, Kayao Lau,Gerburg Wulf,Aditya Bardia,Laura Spring,Steven Isakoff,Jochen Lennerz,Levi Pierce,Ermira Pazolli,Gad Getz,Ryan Corcoran,Dejan Juric Cancer Research(2024)
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