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Fit-for-Purpose Synthesis of a KRASG12C Covalent Inhibitor, Via a Diastereoselective Hayashi Arylation

ORGANIC PROCESS RESEARCH & DEVELOPMENT(2024)

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关键词
KRAS(G12C),Hayashi arylation,asymmetricmonohydrogenation of 1,4-dienes,SimplePHOX
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