Development of a Sensitive High-throughput Enzymatic Assay Capable of Measuring Sub-nanomolar Inhibitors of SARS-CoV2 Mpro
SLAS DISCOVERY(2024)
关键词
Enzyme assays,Enzyme kinetics,SARS-CoV-2 main protease (Mpro),Positive cooperativity,Kosmotropic anion salts,Dimer-monomer equilibrium
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