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The Study of Halogen Effect on the Reactivity of the Serine-Targeting Covalent Warheads

Conghao Gai, Ya Zhang, Shihao Zhang, Xueyan Hu, Yun-Qing Song, Xiaoyu Zhuang,Xiaoyun Chai,Yan Zou,Guang-Bo Ge,Qingjie Zhao

FRONTIERS IN CHEMISTRY(2024)

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关键词
hCES1A,covalent warheads,2,2,2-trifluoroacetophenones,serine-targeted reactivity,halogen effect
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