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Unlocking the Antiviral Arsenal: Structure-Guided Optimization of Small-Molecule Inhibitors Against RSV and Hcov-229E

Christina Karhan,Svenja M. Sake,Antonia P. Gunesch,Christina Grethe, Benedikt Hellwinkel, Natalie M. Köhler,Alexander F. Kiefer, Uladzislau Hapko,Andreas M. Kany,Thomas Pietschmann,Anna K.H. Hirsch

European Journal of Medicinal Chemistry(2025)

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关键词
RSV inhibitors,hCoV-229E inhibitors,Structure-guided optimization,SAR,Selectivity,Small molecules
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