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Identification of Structurally Novel KRASG12C Inhibitors Through Covalent DNA-Encoded Library Screening

David Huang, Francesco Manoni, Zhen Sun, Rongfeng Liu,Jennifer R. Allen, Abhisek Banerjee,Victor J. Cee, Josephine Eshon,Michael J. Frohn,Matthew R. Kaller, Heejun Lee, Cui Li,Xun Li,Patricia Lopez,Vu Ma, Jose M. Medina,Christopher Mohr, Olga A. Mukhina,Alexander J. Pickrell, John Stellwagen, Wenting Wu, Wenhan Zhang, Kai Zhu,Upendra P. Dahal,Liaoyuan A. Hu, Monica Leavitt, Wencui Li, Yu Li,Yingli Ma,Karen Rex,Anne Y. Saiki,Paul Wang, Yaping Sun,Dongcheng Dai,Nuria A. Tamayo,Brian A. Lanman

JOURNAL OF MEDICINAL CHEMISTRY(2025)

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